Synthesis and antitubercular activity of imidazo [2, 1-b] thiazoles A Andreani, M Granaiola, A Leoni, A Locatelli, R Morigi, M Rambaldi European Journal of Medicinal Chemistry 36 (9), 743-746, 2001 | 203 | 2001 |
New Antitumor Imidazo[2,1-b]thiazole Guanylhydrazones and Analogues1 A Andreani, S Burnelli, M Granaiola, A Leoni, A Locatelli, R Morigi, ... Journal of medicinal chemistry 51 (4), 809-816, 2008 | 176 | 2008 |
New isatin derivatives with antioxidant activity A Andreani, S Burnelli, M Granaiola, A Leoni, A Locatelli, R Morigi, ... European journal of medicinal chemistry 45 (4), 1374-1378, 2010 | 144 | 2010 |
Antitumor activity of bis-indole derivatives A Andreani, S Burnelli, M Granaiola, A Leoni, A Locatelli, R Morigi, ... Journal of medicinal chemistry 51 (15), 4563-4570, 2008 | 143 | 2008 |
Imidazo[2,1-b]thiazole System: A Scaffold Endowing Dihydropyridines with Selective Cardiodepressant Activity R Budriesi, P Ioan, A Locatelli, S Cosconati, A Leoni, MP Ugenti, ... Journal of medicinal chemistry 51 (6), 1592-1600, 2008 | 107 | 2008 |
Potential antitumor agents. Part 291: synthesis and potential coanthracyclinic activity of imidazo [2, 1-b] thiazole guanylhydrazones A Andreani, A Leoni, A Locatelli, R Morigi, M Rambaldi, M Recanatini, ... Bioorganic & medicinal chemistry 8 (9), 2359-2366, 2000 | 104 | 2000 |
Potential Antitumor Agents. 37. Synthesis and Antitumor Activity of Guanylhydrazones from Imidazo[2,1-b]thiazoles and from the New Heterocyclic System Thiazolo[2¡,3¡:2,3 … A Andreani, M Granaiola, A Leoni, A Locatelli, R Morigi, M Rambaldi, ... Journal of medicinal chemistry 48 (8), 3085-3089, 2005 | 96 | 2005 |
Imidazo [2, 1-b] thiazole guanylhydrazones as RSK2 inhibitors A Andreani, M Granaiola, A Leoni, A Locatelli, R Morigi, M Rambaldi, ... European journal of medicinal chemistry 46 (9), 4311-4323, 2011 | 90 | 2011 |
Synthesis and antitumor activity of substituted 3‐(5‐imidazo [2, 1‐b] thiazolylmethylene)‐2‐indolinones A Andreani, M Granaiola, A Leoni, A Locatelli, R Morigi, M Rambaldi, ... Anti-cancer drug design 16 (2), 167-174, 2001 | 80 | 2001 |
Antitumor Activity of Substituted E-3-(3,4,5-Trimethoxybenzylidene)-1,3-dihydroindol-2-ones A Andreani, S Burnelli, M Granaiola, A Leoni, A Locatelli, R Morigi, ... Journal of medicinal chemistry 49 (23), 6922-6924, 2006 | 79 | 2006 |
Substituted 3-(5-Imidazo[2,1-b]thiazolylmethylene)-2-indolinones and Analogues: Synthesis, Cytotoxic Activity, and Study of the Mechanism of Action A Andreani, M Granaiola, A Locatelli, R Morigi, M Rambaldi, L Varoli, ... Journal of Medicinal Chemistry 55 (5), 2078-2088, 2012 | 78 | 2012 |
Antitumor Activity of New Substituted 3-(5-Imidazo[2,1-b]thiazolylmethylene)-2-indolinones and 3-(5-Imidazo[2,1-b]thiadiazolylmethylene)-2-indolinones … A Andreani, S Burnelli, M Granaiola, A Leoni, A Locatelli, R Morigi, ... Journal of medicinal chemistry 51 (23), 7508-7513, 2008 | 78 | 2008 |
Synthesis and cardiotonic activity of imidazo [2, lb] thiazoles bearing a lactam ring A Andreani, M Rambaldi, A Leoni, A Locatelli, R Bossa, M Chiericozzi, ... European journal of medicinal chemistry 31 (5), 383-387, 1996 | 78 | 1996 |
Recent patents on thiazole derivatives endowed with antitumor activity R Morigi, A Locatelli, A Leoni, M Rambaldi Recent patents on anti-cancer drug discovery 10 (3), 280-297, 2015 | 76 | 2015 |
Novel thiazole derivatives: a patent review (2008–2012; Part 1) A Leoni, A Locatelli, R Morigi, M Rambaldi Expert opinion on therapeutic patents 24 (2), 201-216, 2014 | 76 | 2014 |
Synthesis and screening for antiacetylcholinesterase activity of (1-benzyl-4-oxopiperidin-3-ylidene) methylindoles and-pyrroles related to donepezil A Andreani, A Cavalli, M Granaiola, M Guardigli, A Leoni, A Locatelli, ... Journal of medicinal chemistry 44 (23), 4011-4014, 2001 | 75 | 2001 |
Synthesis of lactams with potential cardiotonic activity A Andreani, M Rambaldi, A Locatelli, A Leoni, R Bossa, M Chiericozzi European journal of medicinal chemistry 28 (10), 825-829, 1993 | 73 | 1993 |
Chemiluminescent high-throughput microassay applied to imidazo [2, 1-b] thiazole derivatives as potential acetylcholinesterase and butyrylcholinesterase inhibitors A Andreani, S Burnelli, M Granaiola, M Guardigli, A Leoni, A Locatelli, ... European journal of medicinal chemistry 43 (3), 657-661, 2008 | 70 | 2008 |
Antitumor Activity of New Substituted 3-(5-Imidazo[2,1-b]thiazolylmethylene)-2-indolinones and Study of Their Effect on the Cell Cycle A Andreani, M Granaiola, A Leoni, A Locatelli, R Morigi, M Rambaldi, ... Journal of medicinal chemistry 48 (17), 5604-5607, 2005 | 69 | 2005 |
Novel thiazole derivatives: a patent review (2008–2012. Part 2) A Leoni, A Locatelli, R Morigi, M Rambaldi Expert opinion on therapeutic patents 24 (7), 759-777, 2014 | 66 | 2014 |