Athanasios Papakyriakou
Athanasios Papakyriakou
Institute of Biosciences and Applications, NCSR "Demokritos"
Verified email at bio.demokritos.gr - Homepage
TitleCited byYear
Dietary flavonoids in cancer therapy and prevention: substrates and inhibitors of cytochrome P450 CYP1 enzymes
VP Androutsopoulos, A Papakyriakou, D Vourloumis, AM Tsatsakis, ...
Pharmacology & therapeutics 126 (1), 9-20, 2010
1742010
The internal sequence of the peptide-substrate determines its N-terminus trimming by ERAP1
I Evnouchidou, F Momburg, A Papakyriakou, A Chroni, L Leondiadis, ...
PLoS One 3 (11), e3658, 2008
892008
Mononuclear metal complexes with Piroxicam: Synthesis, structure and biological activity
P Christofis, M Katsarou, A Papakyriakou, Y Sanakis, N Katsaros, ...
Journal of inorganic biochemistry 99 (11), 2197-2210, 2005
812005
Comparative CYP1A1 and CYP1B1 substrate and inhibitor profile of dietary flavonoids
VP Androutsopoulos, A Papakyriakou, D Vourloumis, DA Spandidos
Bioorganic & medicinal chemistry 19 (9), 2842-2849, 2011
772011
Probing the S1 specificity pocket of the aminopeptidases that generate antigenic peptides
E Zervoudi, A Papakyriakou, D Georgiadou, I Evnouchidou, A Gajda, ...
Biochemical Journal 435 (2), 411-420, 2011
672011
A common single nucleotide polymorphism in endoplasmic reticulum aminopeptidase 2 induces a specificity switch that leads to altered antigen processing
I Evnouchidou, J Birtley, S Seregin, A Papakyriakou, E Zervoudi, ...
The Journal of Immunology 189 (5), 2383-2392, 2012
582012
Anticancer effects of the metabolic products of the resveratrol analogue, DMU-212: structural requirements for potency
VP Androutsopoulos, KC Ruparelia, A Papakyriakou, H Filippakis, ...
European journal of medicinal chemistry 46 (6), 2586-2595, 2011
542011
Pyrrolo[2,3-a]carbazoles as Potential Cyclin Dependent Kinase 1 (CDK1) Inhibitors. Synthesis, Biological Evaluation, and Binding Mode through Docking Simulations
MA Fousteris, A Papakyriakou, A Koutsourea, M Manioudaki, ...
Journal of medicinal chemistry 51 (4), 1048-1052, 2008
492008
A new role for Zn (II) aminopeptidases: antigenic peptide generation and destruction
I Evnouchidou, A Papakyriakou, E Stratikos
Current pharmaceutical design 15 (31), 3656-3670, 2009
442009
Effects of polymorphic variation on the mechanism of Endoplasmic Reticulum Aminopeptidase 1
A Stamogiannos, D Koumantou, A Papakyriakou, E Stratikos
Molecular immunology 67 (2), 426-435, 2015
332015
Synthesis and biopharmaceutical evaluation of imatinib analogues featuring unusual structural motifs
KC Nicolaou, D Vourloumis, S Totokotsopoulos, A Papakyriakou, ...
ChemMedChem 11 (1), 31-37, 2016
312016
Molecular interaction of α-conotoxin RgIA with the rat α9α10 nicotinic acetylcholine receptor
L Azam, A Papakyriakou, M Zouridakis, P Giastas, SJ Tzartos, ...
Molecular pharmacology 87 (5), 855-864, 2015
312015
Conformational dynamics of the EGFR kinase domain reveals structural features involved in activation
A Papakyriakou, D Vourloumis, F Tzortzatou‐Stathopoulou, M Karpusas
Proteins: Structure, Function, and Bioinformatics 76 (2), 375-386, 2009
312009
Simulated interactions between angiotensin-converting enzyme and substrate gonadotropin-releasing hormone: novel insights into domain selectivity
A Papakyriakou, GA Spyroulias, ED Sturrock, E Manessi-Zoupa, ...
Biochemistry 46 (30), 8753-8765, 2007
292007
Synthesis and Structures of Se Analogues of the Antithyroid Drug 6‐n‐Propyl‐2‐thiouracil and Its Alkyl Derivatives: Formation of Dimeric Se–Se Compounds and …
CD Antoniadis, SK Hadjikakou, N Hadjiliadis, A Papakyriakou, M Baril, ...
Chemistry–A European Journal 12 (26), 6888-6897, 2006
282006
Synthesis of bicyclic molecular scaffolds (BTAa): an investigation towards new selective MMP-12 inhibitors
C Mannino, M Nievo, F Machetti, A Papakyriakou, V Calderone, M Fragai, ...
Bioorganic & medicinal chemistry 14 (22), 7392-7403, 2006
262006
Study of the inclusion of the (R)-and (S)-camphor enantiomers in α-cyclodextrin by X-ray crystallography and molecular dynamics
A Kokkinou, F Tsorteki, M Karpusas, A Papakyriakou, K Bethanis, ...
Carbohydrate research 345 (8), 1034-1040, 2010
212010
A computational approach to the study of the binding mode of dual ACE/NEP inhibitors
N Dimitropoulos, A Papakyriakou, GA Dalkas, ED Sturrock, GA Spyroulias
Journal of chemical information and modeling 50 (3), 388-396, 2010
202010
Optimization and structure–activity relationships of phosphinic pseudotripeptide inhibitors of aminopeptidases that generate antigenic peptides
P Kokkala, A Mpakali, FX Mauvais, A Papakyriakou, I Daskalaki, ...
Journal of medicinal chemistry 59 (19), 9107-9123, 2016
192016
Low molecular weight inhibitors of the protease anthrax lethal factor
GA Dalkas, A Papakyriakou, A Vlamis-Gardikas, GA Spyroulias
Mini reviews in medicinal chemistry 8 (3), 290, 2008
192008
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