Andrea Brancale
Andrea Brancale
Verified email at cardiff.ac.uk
TitleCited byYear
New arylthioindoles: Potent Inhibitors of tubulin polymerization. 2. Structure− activity relationships and molecular modeling studies
G De Martino, MC Edler, G La Regina, A Coluccia, MC Barbera, D Barrow, ...
Journal of medicinal chemistry 49 (3), 947-954, 2006
3352006
Indole, a core nucleus for potent inhibitors of tubulin polymerization
A Brancale, R Silvestri
Medicinal research reviews 27 (2), 209-238, 2007
3082007
Arylthioindoles, potent inhibitors of tubulin polymerization
G De Martino, G La Regina, A Coluccia, MC Edler, MC Barbera, ...
Journal of medicinal chemistry 47 (25), 6120-6123, 2004
2342004
Potent and selective inhibition of varicella-zoster virus (VZV) by nucleoside analogues with an unusual bicyclic base
C McGuigan, CJ Yarnold, G Jones, S Velázquez, H Barucki, A Brancale, ...
Journal of medicinal chemistry 42 (22), 4479-4484, 1999
2291999
Arylthioindole inhibitors of tubulin polymerization. 3. Biological evaluation, structure− activity relationships and molecular modeling studies
G La Regina, MC Edler, A Brancale, S Kandil, A Coluccia, F Piscitelli, ...
Journal of medicinal chemistry 50 (12), 2865-2874, 2007
1492007
Synthesis and antitumor activity of 1, 5-disubstituted 1, 2, 4-triazoles as cis-restricted combretastatin analogues
R Romagnoli, PG Baraldi, O Cruz-Lopez, C Lopez Cara, MD Carrion, ...
Journal of medicinal chemistry 53 (10), 4248-4258, 2010
1442010
Synthesis and evaluation of 1, 5-disubstituted tetrazoles as rigid analogues of combretastatin A-4 with potent antiproliferative and antitumor activity
R Romagnoli, PG Baraldi, MK Salvador, D Preti, M Aghazadeh Tabrizi, ...
Journal of medicinal chemistry 55 (1), 475-488, 2011
1322011
Design, synthesis, and biological evaluation of thiophene analogues of chalcones
R Romagnoli, PG Baraldi, MD Carrion, CL Cara, O Cruz-Lopez, D Preti, ...
Bioorganic & medicinal chemistry 16 (10), 5367-5376, 2008
1322008
Synthesis and biological evaluation of 2-and 3-aminobenzo [b] thiophene derivatives as antimitotic agents and inhibitors of tubulin polymerization
R Romagnoli, PG Baraldi, MD Carrion, CL Cara, D Preti, F Fruttarolo, ...
Journal of medicinal chemistry 50 (9), 2273-2277, 2007
1242007
Indolylarylsulfones as HIV-1 non-nucleoside reverse transcriptase inhibitors: new cyclic substituents at indole-2-carboxamide
G La Regina, A Coluccia, A Brancale, F Piscitelli, V Gatti, G Maga, ...
Journal of medicinal chemistry 54 (6), 1587-1598, 2011
121*2011
Exploring the structural requirements for inhibition of the ubiquitin E3 ligase breast cancer associated protein 2 (BCA2) as a treatment for breast cancer
G Brahemi, FR Kona, A Fiasella, D Buac, J Soukupová, A Brancale, ...
Journal of medicinal chemistry 53 (7), 2757-2765, 2010
1072010
Design, synthesis and evaluation of a novel double pro-drug: INX-08189. A new clinical candidate for hepatitis C virus
C McGuigan, K Madela, M Aljarah, A Gilles, A Brancale, N Zonta, ...
Bioorganic & medicinal chemistry letters 20 (16), 4850-4854, 2010
982010
The tubulin colchicine domain: a molecular modeling perspective
A Massarotti, A Coluccia, R Silvestri, G Sorba, A Brancale
ChemMedChem 7 (1), 33-42, 2012
952012
Synthesis and biological evaluation of 1-methyl-2-(3′, 4′, 5′-trimethoxybenzoyl)-3-aminoindoles as a new class of antimitotic agents and tubulin inhibitors
R Romagnoli, PG Baraldi, T Sarkar, MD Carrion, CL Cara, O Cruz-Lopez, ...
Journal of medicinal chemistry 51 (5), 1464-1468, 2008
912008
New arylthioindoles and related bioisosteres at the sulfur bridging group. 4. Synthesis, tubulin polymerization, cell growth inhibition, and molecular modeling studies
G La Regina, T Sarkar, R Bai, MC Edler, R Saletti, A Coluccia, F Piscitelli, ...
Journal of medicinal chemistry 52 (23), 7512-7527, 2009
892009
Toward highly potent cancer agents by modulating the C-2 group of the arylthioindole class of tubulin polymerization inhibitors
G La Regina, R Bai, WM Rensen, E Di Cesare, A Coluccia, F Piscitelli, ...
Journal of medicinal chemistry 56 (1), 123-149, 2012
882012
Convergent synthesis and biological evaluation of 2-amino-4-(3′, 4′, 5′-trimethoxyphenyl)-5-aryl thiazoles as microtubule targeting agents
R Romagnoli, PG Baraldi, A Brancale, A Ricci, E Hamel, R Bortolozzi, ...
Journal of medicinal chemistry 54 (14), 5144-5153, 2011
752011
The application of phosphoramidate protide technology to acyclovir confers anti-HIV inhibition
M Derudas, D Carta, A Brancale, C Vanpouille, A Lisco, L Margolis, ...
Journal of medicinal chemistry 52 (17), 5520-5530, 2009
722009
Design, synthesis and structure–activity relationship of 2-(3′, 4′, 5′-trimethoxybenzoyl)-benzo [b] furan derivatives as a novel class of inhibitors of tubulin polymerization
R Romagnoli, PG Baraldi, MD Carrion, CL Cara, O Cruz-Lopez, ...
Bioorganic & medicinal chemistry 17 (19), 6862-6871, 2009
702009
Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus
M Bassetto, T De Burghgraeve, L Delang, A Massarotti, A Coluccia, ...
Antiviral research 98 (1), 12-18, 2013
692013
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